
Discovery Program
We are actively exploring additional opportunities to leverage our pan-variant targeted therapy approach to address treatment resistant cancers.
Our structure-guided drug design approach, integrated with our predictive resistance assay (PRA), allows us to efficiently design and validate novel inhibitors that target all major activating and resistance mutations for a given target. We are currently evaluating several potential targets for a next-generation inhibitor against a clinically validated driver oncogene.
We intend to nominate at least one of these inhibitors as our next program in 2022.

We are developing a pipeline of TKIs designed to inhibit all major cancer causing and drug resistance mutations in clinically significant protein kinases.
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